Sitaxentan

Scheme

Rec.INN

ATC (Anatomical Therapeutic Chemical Classification)

C02KX03

CAS registry number (Chemical Abstracts Service)

0184036-34-8

Chemical Formula

C18-H15-Cl-N2-O6-S2

Molecular Weight

454

Therapeutic Category

Endothelin antagonist

Chemical Names

N-(4-Chlor-3-methylisoxazol-5-yl)-2-[(4,5-methylendioxy-2-methylphenyl)acetyl]thiophen-3-sulfonamid (IUPAC)

N-(4-Chlor-3-methylisoxazol-5-yl)-2-[2-(6-methyl-1,3-benzodioxol-5-yl)acetyl]thiophen-3-sulfonamid

N-(4-Chloro-3-methyl-5-isoxazolyl)-2-[[4,5-(methylenedioxy)-o-tolyl]acetyl]-3-thiophenesulfonamide (WHO)

3-Thiophenesulfonamide, N-(4-chloro-3-methyl-5-isoxazolyl)-2-[[6-methyl-1,3-benzodioxol-5-yl]acetyl]-

Foreign Names

• Sitaxentanum (Latin)
• Sitaxentan (German)
• Sitaxentan (French)
• Sitaxentan (Spanish)

Generic Names

• IPI 1040 (IS)
• Sitaxsentan (IS)
• LGLS (IS)
• TBC-11241 (IS)
• TBC-11251 (IS: TexasBiotechn)
• TBC-2576 (IS)
• TBC-3214 (IS)

Brand Names

• Thelin
  Praxis Pharmaceutical, Spain; CSL, Australia; Encysive, Austria; Encysive, Germany; Encysive, France; Encysive, United Kingdom; Encysive, Ireland; Encysive, Luxembourg; Encysive, Netherlands; LCA, Belgium; EncysiveUK Limited, Denmark



• THELIN
  Pfizer, Sweden

International Drug Name Search

Glossary

IUPAC	International Union of Pure and Applied Chemistry
IS	Inofficial Synonym
Rec.INN	Recommended International Nonproprietary Name (World Health Organization)
WHO	World Health Organization

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